Release modulator
A release modulator, or neurotransmitter release modulator, is a type of drug that modulates the release of one or more neurotransmitters. Examples of release modulators include monoamine releasing agents such as the substituted amphetamines (which induce the release of norepinephrine, dopamine, and/or serotonin) and release inhibitors such as botulinum toxin A (which inhibits acetylcholine release by inactivating SNAP-25, thereby preventing exocytosis from occurring).
See also
References
|
---|
Amino acids and similar/related |
- Amino acids and related: GABA receptor modulators
- GABAA receptor positive allosteric modulators
- GHB receptor modulators
- Glutamate receptor modulators
- Glycine receptor modulators
- Monoamines: Adrenergic receptor modulators
- Dopamine receptor modulators
- Histamine receptor modulators
- Melatonin receptor modulators
- Monoamine metabolism modulators
- Monoamine neurotoxins
- Monoamine releasing agents
- Monoamine reuptake inhibitors
- Serotonin receptor modulators
- TAAR modulators
- Others: Acetylcholine receptor modulators
- Imidazoline receptor modulators
- Purine receptor modulators
- Sigma receptor modulators
- Thyroid hormone receptor modulators
|
---|
Lipids |
- Eicosanoids: Cannabinoid receptor modulators
- Leukotriene signaling modulators
- Prostanoid signaling modulators
- Phospholipids: Lysophospholipid signaling modulators
- PAF receptor modulators
- Steroids and related: Androgen receptor modulators
- Estrogen receptor modulators
- Glucocorticoid receptor modulators
- Mineralocorticoid receptor modulators
- Nuclear receptor modulators
- Progesterone receptor modulators
- Steroid metabolism modulators
|
---|
Peptides/proteins |
- General: Signaling peptide/protein receptor modulators
- Peptides: GH/IGF-1 axis signaling modulators
- Melanocortin receptor modulators
- Opioid receptor modulators
- Oxytocin and vasopressin receptor modulators
- Cytokines: Cytokine receptor modulators
- Chemokine receptor modulators
- Interleukin receptor modulators
- TNF receptor superfamily modulators
- Growth factors: Growth factor receptor modulators
- TGFβ receptor superfamily modulators
|
---|
Others and non-receptor |
- Ion channels: Ion channel modulators
- TRP channel modulators
- Transporters: Symporter inhibitors
- Others: Nitric oxide signaling modulators
|
---|
- See also
- Pharmacomodulation
- Cell signaling
- Neurotransmitters
|
|
---|
Types | |
---|
Classes | | see Enzyme inhibition |
---|
| |
---|
| |
---|
Miscellaneous | |
---|
|
---|