List of estrogen esters

Estradiol, the base estrogen of most estrogen esters.

This is a list of estrogen esters, including esters (as well as ethers) of steroidal estrogens like estradiol, estrone, and estriol and nonsteroidal estrogens like the stilbestrols diethylstilbestrol and hexestrol.

Esters of steroidal estrogens

Estradiol esters

Marketed

Many esters of estradiol have been marketed, including the following major esters:[1][2]

And the following less commonly used esters:[1][2]

The following nitrogen mustard ester of estradiol is an alkylating antineoplastic agent and has been marketed:[1][2]

Never marketed

A few other estradiol esters which are notable but have not been marketed include:[2]

The following alkylating antineoplastic nitrogen mustard esters of estradiol have not been marketed:[2]

Estrone esters

Marketed

Esters of estrone that have been marketed include:[1][2]

Never marketed

Other estrone esters which are notable but have not been marketed include:

Estriol esters

Marketed

Esters of estriol that have been marketed include:[1][2]

Never marketed

The following ester of estriol was never marketed:

Esters of other steroidal estrogens

Marketed

The following esters of other estrogens exist and have been marketed:[1]

Ethers of steroidal estrogens

Marketed

A number of estrogen ethers also exist and have been marketed, including:[5][1]

Never marketed

A few other estrogen ethers which are notable but have not been marketed include:[5]

Esters of nonsteroidal estrogens

Diethylstilbestrol esters

Marketed

Major esters of diethylstilbestrol include:

Less commonly used esters of diethylstilbestrol include:

Never marketed

As well as the following nitrogen mustard ester:

Hexestrol esters

Marketed

Never marketed

The following nitrogen mustard ester of hexestrol was never marketed:

Esters of other nonsteroidal estrogens

Marketed

Ethers of nonsteroidal estrogens

Diethylstilbestrol

Marketed

See also

References

  1. 1 2 3 4 5 6 7 Index Nominum 2000: International Drug Directory. Taylor & Francis US. 2000. p. 404. ISBN 978-3-88763-075-1. Retrieved 29 May 2012.
  2. 1 2 3 4 5 6 7 A. D. Roberts (1991). Dictionary of Steroids: Chemical Data, Structures, and Bibliographies. CRC Press. p. 415. ISBN 978-0-412-27060-4. Retrieved 20 May 2012.
  3. ↑ Dahlgren E, Crona N, Janson PO, Samsioe G (1985). "Oral replacement with estradiol-cyclooctyl acetate: a new estradiol analogue. Effects on serum lipids, proteins, gonadotrophins, estrogens and uterine endometrial morphology". Gynecol. Obstet. Invest. 20 (2): 84–90. PMID 3932144.
  4. ↑ Luisi M, Kicovic PM, Alicicco E, Franchi F (1978). "Effects of estradiol decanoate in ovariectomized women". J. Endocrinol. Invest. 1 (2): 101–6. PMID 755846. doi:10.1007/BF03350355.
  5. 1 2 J. Elks (14 November 2014). The Dictionary of Drugs: Chemical Data: Chemical Data, Structures and Bibliographies. Springer. ISBN 978-1-4757-2085-3.
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