Levophenacylmorphan
Systematic (IUPAC) name | |
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(−)-3-Hydroxy-N-phenacylmorphinan | |
Clinical data | |
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Identifiers | |
10061-32-2 | |
None | |
PubChem | CID 5362482 |
ChemSpider | 16736786 |
UNII | 7Q24AL2BR2 |
Synonyms | Levophenacylmorphan |
Chemical data | |
Formula | C24H27NO2 |
361.48 g/mol | |
SMILES
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Levophenacylmorphan is a morphinan derivative that acts as an opioid agonist. It has potent analgesic effects and is around 10x more potent than morphine.[1] Adverse effects associated with its use are those of the opioids as a whole, including pruritus, nausea, respiratory depression, euphoria and development of tolerance and dependence to its effects.[2]
References
- ↑ MAY, E.L. & EDDY, N.B., A New Potent Synthetic Analgesic, J. Org. Chem., 24 : 294, 1959.
- ↑ Fraser HF, Isbell H. Human pharmacology and addiction liabilities of phenazocine and levophenacylmorphan. UN Bulletin on Narcotics. 1960 Issue 2