Oxetorone

Oxetorone
Systematic (IUPAC) name
(3Z)-3-[1]benzofuro[3,2-c][1]benzoxepin-6(12H)-ylidene-N,N-dimethylpropan-1-amine
Clinical data
AHFS/Drugs.com International Drug Names
Pregnancy cat.  ?
Legal status  ?
Identifiers
CAS number 26020-55-3 Y
ATC code N02CX06
PubChem CID 6436540
UNII T3XOS33TIQ Y
KEGG D08312 Y
Chemical data
Formula C21H21NO2 
Mol. mass 319.40 g/mol
SMILES eMolecules & PubChem
 Y(what is this?)  (verify)

Oxetorone is an antimigraine agent.[1]

Association with hyperprolactinemia has been described.[2]

References

  1. ^ Massiou H (2000). "[Prophylactic treatments of migraine"] (in French). Rev. Neurol. (Paris) 156 Suppl 4: 4S79–86. PMID 11139754. http://www.masson.fr/masson/79997. 
  2. ^ Pradalier A (December 1996). "Hyperprolactinaemia and depression induced by oxetorone". Cephalalgia 16 (8): 560–1. doi:10.1046/j.1468-2982.1996.1608560.x. PMID 8980859. http://www3.interscience.wiley.com/resolve/openurl?genre=article&sid=nlm:pubmed&issn=0333-1024&date=1996&volume=16&issue=8&spage=560. 
Antimigraine preparations (N02C)
Analgesic/abortive
Serotonin modulators
Ergot alkaloids
Other
Other
Prevention of migraines
Ungrouped
Pizotifen • Iprazochrome • Dimetotiazine • Oxetorone • Lomerizine • Telcagepant

M: CNS

anat(n/s/m/p/4/e/b/d/c/a/f/l/g)/phys/devp

noco(m/d/e/h/v/s)/cong/tumr, sysi/epon, injr

proc, drug(N1A/2AB/C/3/4/7A/B/C/D)