Epelsiban

Epelsiban
Systematic (IUPAC) name
(3R,6R)-3-(2,3-dihydro-1H-inden-2-yl)-1-[(1R)-1-(2,6-dimethylpyridin-3-yl)-2-(morpholin-4-yl)-2-oxoethyl]-6-[(1S)-1-methylpropyl]piperazine-2,5-dione
Clinical data
Pregnancy cat.  ?
Legal status Non-regulated
Identifiers
CAS number 872599-83-2
1159097-48-9 (besylate)
ATC code None
Chemical data
Formula C30H38N4O4 
Mol. mass 518.6 g/mol

Epelsiban (GSK-557,296-B) is a drug which acts as an non-peptide oxytocin receptor antagonist, and is being developed by GlaxoSmithKline for the treatment of premature ejaculation in men.[1][2]

See also

References