Regadenoson
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Regadenoson
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Systematic (IUPAC) name | |
1-[6-amino-9-[(2R,3R,4S,5R)-3,4-dihydroxy-5- (hydroxymethyl)oxolan-2-yl]purin-2-yl]- N-methylpyrazole-4-carboxamide | |
Identifiers | |
CAS number | 875148-45-1 |
ATC code | ? |
PubChem | |
Chemical data | |
Formula | C15H18N8O5 |
Mol. mass | 390.354 g/mol |
Synonyms | 2-[4-[(methylamino)carbonyl]- 1H-pyrazol-1-yl]-adenosine |
Pharmacokinetic data | |
Bioavailability | ? |
Metabolism | ? |
Half life | ? |
Excretion | ? |
Therapeutic considerations | |
Licence data |
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Pregnancy cat. |
C(US) |
Legal status | |
Routes | Intravenous |
Regadenoson (INN, codenamed CVT-3146) is an A2A adenosine receptor agonist that is a coronary vasodilator.
It was approved by the United States Food and Drug Administration on April 10, 2008 and it will be marketed under the tradename Lexiscan.[1] It has not yet gained approval in the European Union.