Regadenoson

From Wikipedia, the free encyclopedia

Regadenoson
Systematic (IUPAC) name
1-[6-amino-9-[(2R,3R,4S,5R)-3,4-dihydroxy-5- (hydroxymethyl)oxolan-2-yl]purin-2-yl]- N-methylpyrazole-4-carboxamide
Identifiers
CAS number 313348-27-5
875148-45-1
ATC code  ?
PubChem 219024
Chemical data
Formula C15H18N8O5 
Mol. mass 390.354 g/mol
Synonyms 2-[4-[(methylamino)carbonyl]- 1H-pyrazol-1-yl]-adenosine
Pharmacokinetic data
Bioavailability  ?
Metabolism  ?
Half life  ?
Excretion  ?
Therapeutic considerations
Licence data

US

Pregnancy cat.

C(US)

Legal status

-only(US)

Routes Intravenous

Regadenoson (INN, codenamed CVT-3146) is an A2A adenosine receptor agonist that is a coronary vasodilator.

It was approved by the United States Food and Drug Administration on April 10, 2008 and it will be marketed under the tradename Lexiscan.[1] It has not yet gained approval in the European Union.

[edit] References