Nalorphine

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Nalorphine
Systematic (IUPAC) name
(−)−(5R,6S)-9α-allyl-4,5-epoxymorphin-7-en-3,6-diol
Identifiers
CAS number 62-67-9
ATC code V03AB02
PubChem 5284595
Chemical data
Formula C19H21NO3 
Mol. mass 311.375 g/mol
Pharmacokinetic data
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Therapeutic considerations
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Legal status
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Nalorphine (INN, also known as N-allyl-normorphine) trade names Lethidrone and Nalline. Nalorphine acts at two opioid receptors, at the mu receptor it has antagonistic effects and at the kappa receptors it exerts agonistic characteristics. It is used to reverse opioid overdose and in a challenge test to determine opioid dependence.

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