Mibolerone

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Mibolerone
Systematic (IUPAC) name
(7R,8R,9S,10R,13S,14S,17S)-17-Hydroxy- 7,13,17-trimethyl-1,2,6,7,8,9,10,11,1

2,14,15,16-dodecahydrocyclopenta[a]phenanthren-3-one

Identifiers
CAS number 3704-09-4
ATC code  ?
PubChem 251636
Chemical data
Formula C20H30O2 
Mol. mass 302.4558 g/mol
Pharmacokinetic data
Bioavailability  ?
Metabolism Hepatic
Half life 2-4 hours
Excretion  ?
Therapeutic considerations
Pregnancy cat.

?

Legal status

Schedule 3 (US)

Routes Oral

Mibolerone is a potent anabolic steroid which is both higher affinity[1] and more selective[2] for the androgen receptor than metribolone.

[edit] References

  1. ^ Murthy LR, Johnson MP, Rowley DR, Young CY, Scardino PT, Tindall DJ (1986). "Characterization of steroid receptors in human prostate using mibolerone". Prostate 8 (3): 241–53. PMID 2422638. 
  2. ^ Schilling K, Liao S (1984). "The use of radioactive 7 alpha, 17 alpha-dimethyl-19-nortestosterone (mibolerone) in the assay of androgen receptors". Prostate 5 (6): 581–8. PMID 6333679.