Metribolone
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| Metribolone | |
|---|---|
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| IUPAC name | 17β-17-Hydroxy-17-methyl-estra-4,9,11-trien-3-one |
| Other names | Methyltrienolone, R1881 |
| Identifiers | |
| CAS number | [965-93-5] |
| PubChem | |
| SMILES | CC1(CCC2C1(C=CC3=C4CCC(=O)C=C4CCC23)C)O |
| Properties | |
| Molecular formula | C19H24O2 |
| Molar mass | 284.39266 |
| Except where noted otherwise, data are given for materials in their standard state (at 25 °C, 100 kPa) Infobox disclaimer and references |
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Metribolone, also known as R1881 is a potent non-aromatizable androgen[1] which has also been used as a photoaffinity label for the androgen receptor.[2]
[edit] References
- ^ Bojar H, Maar K, Staib W (1980). "The endocrine background of human renal cell carcinoma. V. Binding of the highly potent androgen methyltrienolone (R 1881) by tumour cytosol". Urol. Int. 35 (2): 154–60. PMID 6966435.
- ^ Brinkmann AO, Kuiper GG, de Boer W, Mulder E, Bolt J, van Steenbrugge GJ, van der Molen HJ (January 1986). "Characterization of androgen receptors after photoaffinity labelling with [3H]methyltrienolone (R1881)". J. Steroid Biochem. 24 (1): 245–9. PMID 2422446.
[edit] External links
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