Bromazine

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Bromazine
Systematic (IUPAC) name
2-[(4-bromophenyl)-phenylmethoxy]-N,N-dimethylethanamine
Identifiers
CAS number 118-23-0
1808-12-4 (hydrochloride)
ATC code R06AA01
PubChem 2444
DrugBank APRD00710
Chemical data
Formula C17H20BrNO 
Mol. mass 334.251 g/mol
SMILES eMolecules & PubChem
Pharmacokinetic data
Bioavailability High
Protein binding 96%
Metabolism Mostly hepatic (CYP-mediated), also renal
Half life 1 to 4 hours
Excretion  ?
Therapeutic considerations
Pregnancy cat.

?

Legal status
Routes Oral

Bromazine (INN, also known as bromodiphenhydramine) is an antihistamine. It is a brominated derivative of diphenhydramine. The medicinal preparation of the hydrochloride has the brand name Ambrodyl