Mibolerone

From Wikipedia, the free encyclopedia

Mibolerone
Systematic (IUPAC) name
(7R,8R,9S,10R,13S,14S,17S)-17-hydroxy- 7,13,17-trimethyl-1,2,6,7,8,9,10,11,1 2,14,15,16-dodecahydrocyclopenta[a]phenanthren-3-one
Identifiers
CAS number	3704-09-4
ATC code	?
PubChem	?
Chemical data
Formula	C20H30O2
Mol. mass	302.4558 g/mol
Pharmacokinetic data
Bioavailability	?
Metabolism	Hepatic
Half life	2-4 hours
Excretion	?
Therapeutic considerations
Pregnancy cat.	?
Legal status	Schedule 3 (US)
Routes	Oral

Mibolerone is an Anabolic steroid which is very androgenic. It is about 5 times more potent than testosterone as an anabolic agent and about 2.5 times more potent as an androgenic agent. It is one of the most androgenic agents in existence and as an effect often causes progesterone related gynecomastia.

v • d • e Sex hormones and related agents (primarily G03, also L02, H01C) - human endogenous in CAPS
Progestogens: (receptor)	PROGESTERONE, Desogestrel, Drospirenone, Dydrogesterone, Ethisterone, Etonogestrel, Ethynodiol diacetate, Gestodene, Gestonorone, Levonorgestrel, Lynestrenol, Medroxyprogesterone, Megestrol, Norelgestromin, Norethisterone, Norethynodrel, Norgestimate, Norgestrel, Norgestrienone, Tibolone Antiprogestogen: Mifepristone
Androgens: (receptor)	TESTOSTERONE, Androstanolone, Fluoxymesterone, Mesterolone, Methyltestosterone, (see also anabolic steroids) Antiandrogens: Bicalutamide, Cyproterone, Flutamide, Nilutamide, Spironolactone
Estrogens: (receptor)	ESTRADIOL, ESTRIOL, ESTRONE, Chlorotrianisene, Dienestrol, Diethylstilbestrol, Ethinylestradiol, Fosfestrol, Mestranol, Polyestradiol phosphate Selective estrogen receptor modulator: Bazedoxifene, Clomifene, Fulvestrant, Raloxifene, Tamoxifen, Toremifene Aromatase inhibitor: Aminogluthetimide, Anastrozole, Exemestane, Formestane, Letrozole, Vorozole
Gonadotropins: (FSHR/LHCGR)	ovulation stim.:Clomifene, Urofollitropin Antigonadotropins: Danazol, Gestrinone
GnRH: (receptor)	agonist: Buserelin, Goserelin, Histrelin, Leuprorelin, Nafarelin, Triptorelin antagonist: Abarelix, Cetrorelix, Ganirelix