Carbetocin

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Carbetocin
Systematic (IUPAC) name
(2S)-1-[(3S,6S,9S,12S,15S)-12-[(2S)-butan-2-yl]-
9-(2-carbamoylethyl)-6-(carbamoylmethyl)-15-
[(4-hydroxyphenyl)methyl]-16-methyl-5,8,11,14,17-
pentaoxo-1-thia-4,7,10,13,16-pentazacycloicosane-
3-carbonyl]-N-[(1S)-1-(carbamoylmethylcarbamoyl)-
3-methyl-butyl]pyrrolidine-2-carboxamide
Identifiers
CAS number 37025-55-1
ATC code H01BB03
PubChem 71715
Chemical data
Formula C45H69N11O12S 
Mol. mass 988.162 g/mol
Pharmacokinetic data
Bioavailability 80% (IM)
Metabolism  ?
Half life 40 minutes
Excretion  ?
Therapeutic considerations
Pregnancy cat.

?

Legal status

POM(UK) Not available (U.S.)

Routes Intravenous, intramuscular

Carbetocin (INN) is a drug used to control postpartum hemorrhage, bleeding after giving birth. It is sold under the trade name Duratocin. It is an analogue of oxytocin, and its action is similar to that of oxytocin; it causes contraction of the uterus.

Carbetocin is available in Canada and the United Kingdom, but not in the United States.

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