Bitolterol

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Image:Bitolterol.png
Bitolterol
Systematic (IUPAC) name
[4-(1-hydroxy-2-tert-butylamino-ethyl)- 2-(4-methylbenzoyl)oxy-phenyl] 4-methylbenzoate
Identifiers
CAS number 30392-41-7
ATC code R03AC17
PubChem 35330
DrugBank APRD00827
Chemical data
Formula C28H31NO5 
Mol. mass 461.549 g/mol
Pharmacokinetic data
Bioavailability  ?
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Therapeutic considerations
Pregnancy cat.

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Legal status
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Bitolterol mesylate (Tornalate®) is a β2-adrenergic receptor agonist used for the relief of bronchospasm in conditions such as asthma and COPD.

Bitolterol has a rapid onset of action (2-5 minutes) and may last up to 6-8 hours.

Bitolterol was withdrawn from the market by Élan Pharmaceuticals in 2001.