Alfentanil

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Alfentanil
Systematic (IUPAC) name
N-[1-[2-(4-ethyl-5-oxo-1,4-dihydrotetrazol-1-yl)ethyl]-
4-(methoxymethyl)-4-piperidyl]-N-phenyl-propanamide
Identifiers
CAS number 71195-58-9
ATC code N01AH02
PubChem 189496
DrugBank APRD00726
Chemical data
Formula C21H32N6O3 
Mol. mass 416.517 g/mol
Physical data
Melt. point 140.8 °C (285 °F)
Pharmacokinetic data
Bioavailability Not applicable
Protein binding 92%
Metabolism Hepatic
Half life 90–111 minutes
Excretion  ?
Therapeutic considerations
Pregnancy cat.

?

Legal status

Schedule II(US)

Routes Intravenous

Alfentanil (trade name Alfenta) is a parenteral short-acting synthetic opioid analgesic drug, used for anaesthesia in surgery. While it gives less cardiovascular complications, it tends to give stronger respiratory depression. Alfentanil is a Schedule II according to the U.S. DEA website.[1]

Alfentanil was discovered at Janssen Pharmaceutica in 1976.

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