Azelastine
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Azelastine
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| Systematic (IUPAC) name | |
| 4-[(4-chlorophenyl)methyl]-2- (1-methylazepan-4-yl)-phthalazin-1-one | |
| Identifiers | |
| CAS number | 58581-89-8 |
| ATC code | R01AC03 R06AX19, S01GX07 |
| PubChem | 2267 |
| DrugBank | APRD00813 |
| Chemical data | |
| Formula | C22H24ClN3O |
| Mol. weight | 381.898 g/mol |
| Pharmacokinetic data | |
| Bioavailability | ? |
| Metabolism | ? |
| Half life | ? |
| Excretion | ? |
| Therapeutic considerations | |
| Pregnancy cat. |
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| Legal status | |
| Routes | ? |
Azelastine is an antihistamine and mast cell stabilizer available as a nasal spray (Astelin®) for hay fever and as eye drops (Optilar®) for allergic conjunctivitis.
[edit] External links
| Antihistamines (primarily R06) edit | ||
|---|---|---|
| Aminoalkyl ethers: |
Bromazine, Carbinoxamine, Clemastine, Chlorphenoxamine, Diphenylpyraline, Diphenhydramine, Doxylamine |
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| Substituted alkylamines: |
Brompheniramine, Chlorphenamine, Dexbrompheniramine , Dexchlorpheniramine, Dimetindene, Pheniramine, Talastine |
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| Substituted ethylene diamines: |
Chloropyramine, Histapyrrodine, Mepyramine, Methapyrilene |
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| Phenothiazine derivatives: |
Alimemazine, Hydroxyethylpromethazine, Isothipendyl, Mequitazine, Methdilazine, Oxomemazine, Promethazine |
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| Piperazine derivatives: |
Buclizine, Cetirizine, Chlorcyclizine, Cinnarizine, Cyclizine, Hydroxyzine, Levocetirizine, Meclozine, Oxatomide |
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| Others for systemic use: |
Acrivastine, Antazoline, Astemizole, Azatadine , Azelastine, Bamipine, Cyproheptadine, Deptropine, Desloratadine, Ebastine, Epinastine, Ketotifen, Loratadine, Mebhydrolin, Mizolastine, Phenindamine, Pimethixene, Pyrrobutamine, Rupatadine, Terfenadine, Triprolidine |
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| For topical use: |
Bamipine, Chloropyramine, Chlorphenoxamine, Clemastine, Dimetindene, Diphenhydramine, Isothipendyl, Mepyramine , Promethazine, Thenalidine |
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| Antiallergic agents excluding corticosteroids: |
Antazoline, Azelastine , Fexofenadine |
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| Other antiallergics: | ||
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